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Annoor Awadasseid

Annoor Awadasseid

LiveDNA ID: 249.41685
15 Publications
0 Editorial Roles
0 Projects

Education

Academic Background
  • Ph.D. University of Chinese Academy of Sciences, Beijing, China Medical Chemistry | Completed: 2020

Publications (15)

Selected Scholarly Contributions
Precision/Locus-Selective G-Quadruplex Stabilization as the Next Medicinal Chemistry Challenge
Jianwei Wang, Haoran Xu, Yuxing Chai, Chenyang Wang, Ping Lv, Koutian Zhang, Yanling Wu, Wen Zhang, Annoor Awadasseid
Journal of Medicinal Chemistry | Journal Article
Crossref
2026
Novel Selenium-Containing Small Molecule PD-L1 Inhibitors: Design, Synthesis, and Evaluation of the Antitumor Activity
Jianwei Wang, Shenwei Yu, Liang Qian, Jacek Plewka, Ruyue Ni, Chenyang Wang, Feng Zhang, Zeyu Chen, Annoor Awadasseid, Yanling Wu, Katarzyna Magiera-Mularz, Wen Zhang
Journal of Medicinal Chemistry | Journal Article
Crossref
2026
Small‐Molecule Inhibitors Targeting PD‐1/PD‐L1 in Colorectal Cancer: Mechanisms, Challenges, and Clinical Prospects
Jianwei Wang, Shenwei Yu, Liang Qian, Yanling Wu, Wen Zhang, Annoor Awadasseid
ChemMedChem | Journal Article
Crossref
2026
Research Progress and Clinical Translation Challenges of Small‐Molecule Inhibitors Targeting PD‐L1
Liang Qian, Ruyue Ni, Ping Lv, Yuxing Chai, Annoor Awadasseid, Xuqiong Xiong, Wen Zhang
ChemMedChem | Journal Article
Crossref
2026
Antiproliferative activity of selenium-enriched coumarin derivatives on the SK-N-SH neuroblastoma cell line: Mechanistic insights
Ming Wang, Haoran Xu, Xuqiong Xiong, Linru Chang, Koutian Zhang, Yongnan Zhou, Feng Zhang, Annoor Awadasseid, Wen Zhang
European Journal of Medicinal Chemistry | Journal Article
Crossref
2025
Advances in cancer immunotherapy using small-molecular inhibitors targeting the PD-1/PD-L1 interaction
Feng Zhang, Sivaramakarthikeyan Ramar, Yu Wang, Haoran Xu, Koutian Zhang, Annoor Awadasseid, Guowu Rao, Wen Zhang
Bioorganic & Medicinal Chemistry | Journal Article
Crossref
2025
Design, Synthesis and Biological Evaluation of Biphenyl-1,2,3-Triazole Hybrid Analogues as PD-1/PD-L1 Inhibitors
Shijia Zhou, Suresh Narva, Mengda Wu, Ming Wang, Feng Zhang, Chenfeng Shen, Annoor Awadasseid, Wen Zhang
International Journal of Pharmacology | Journal Article
Crossref
2024
Design, synthesis, and evaluation of antitumor activity of 2-arylmethoxy-4-(2-fluoromethyl-biphenyl-3-ylmethoxy) benzylamine derivatives as PD-1/PD-l1 inhibitors
Feng Zhang, Hua Zhang, Shijia Zhou, Jacek Plewka, Ming Wang, Shishi Sun, Caiyun Wu, Qimeng Yu, Mengyu Zhu, Annoor Awadasseid, Yanling Wu, Katarzyna Magiera-Mularz, Wen Zhang
European Journal of Medicinal Chemistry | Journal Article
Crossref
2024
Design, synthesis and biological evaluation of novel TMPRSS2-PROTACs with florosubstituted 4-guanidino-N-phenylbenzamide derivative ligands
Hao Yang, Haoran Xu, Xinxin Lin, Zengxuan Cai, Yong Xia, Yu Wang, Zejie Chen, Koutian Zhang, Yanling Wu, Jianwei Wang, Annoor Awadasseid, Wen Zhang
Bioorganic & Medicinal Chemistry | Journal Article
Crossref
2024
Exploring potential bacterial populations for enhanced anthraquinone dyes biodegradation: a critical review
Mayada Jamal, Annoor Awadasseid, Xiaomei Su
Biotechnology Letters | Journal Article
Crossref
2022
Characterization of Camptotheca acuminata 10-hydroxygeraniol oxidoreductase and iridoid synthase and their application in biological preparation of nepetalactol in Escherichia coli featuring NADP+ - NADPH cofactors recycling.
Awadasseid, A., W. Li, Z. Liu, C. Qiao, J. Pang, G. Zhang and Y. Luo,
Int. J. Biol. Macromol., | Journal Article
Self Annoor Awadasseid
2020
Ezrin as a possible diagnostic and/or prognostic biomarker in mice lymphatic metastatic hepatocellular carcinoma in vivo.
Bakheet, A.M.H., S.A. Mahmoud, Y. Huang, J. Zhang and J. Wang et al.,
BioFactors, | Journal Article
Self Annoor Awadasseid
2017
Effect of Coriolus versicolor glucan on the stimulation of cytokine production in sarcoma-180-bearing mice.
Awadasseid, A., K. Eugene, M. Jamal, J. Hou and A.M. Hago, et al.,
Biomed. Rep., | Journal Article
Self Annoor Awadasseid
2017
Lactobacillus rhamnosus induced epithelial cell apoptosis, ameliorates inflammation and prevents colon cancer development in an animal model.
Gamallat, Y., A. Meyiah, E.D. Kuugbee, A.M. Hago and G. Chiwala et al.,
Biomed. Pharmacother., | Journal Article
Self Annoor Awadasseid
2016
Structural change in microbiota by a probiotic cocktail enhances the gut barrier and reduces cancervia TLR2 signaling in a rat model of colon cancer.
Kuugbee, E.D., X. Shang, Y. Gamallat, D. Bamba and A. Awadasseid et al.,
Dig. Dis. Sci., | Journal Article
Self Annoor Awadasseid
2016